SCHEMBL14979306

SCHEMBL14979306

O=c1c(NCCc2ccc(Oc3ccccc3)cc2)c(NC2CCCNC2)c1=O

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FES P07332 1/20 0.51
FGFR1 P11362 1/20 0.51
FLT4 P35916 1/20 0.51
KDR P35968 1/20 0.51
CHEK1 O14757 1/20 0.42
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
POLB P06746 1/20 0.39
BTK Q06187 8/20 0.38
LTA4H P09960 4/20 0.37
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
PLAAT3 P53816 1/20 0.36
PLAAT5 Q96KN8 1/20 0.36
PLAAT2 Q9NWW9 1/20 0.36
PLAAT4 Q9UL19 1/20 0.36
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14979454 0.80 HDAC1 (0.42) CHEK1MEN1KMT2AAURKARPS6KB1
SCHEMBL14979304 0.72 KDM4E (0.46) CHEK1MEN1KMT2A
SCHEMBL10496394 0.69 TAAR1 (0.57) EPHX2
SCHEMBL14813680 0.69 TAAR1 (0.57) EPHX2
SCHEMBL4025807 0.68 FLT4 (1.00) FESFGFR1FLT4KDRCHEK1
SCHEMBL13576621 0.67 EED (0.59) KMT2ALTA4H
SCHEMBL3890476 0.67 EED (0.59) KMT2ALTA4H
SCHEMBL14979456 0.67 HDAC1 (0.41)
SCHEMBL21460332 0.66 MAPT (0.43) CHEK1LTA4H
SCHEMBL4027877 0.65 FES (0.77) FESFGFR1FLT4KDRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8450348-B2 Such as 3-[6-(4-Chloro-phenoxy)-hexylamino]-4-(pyridin-4-ylamino)-cyclobut-3-ene-1,2-dione; cancer, tumors; reduced side effects FORMA TM, LLC (US) 2013-05-28 US disclosed