SCHEMBL1498906

SCHEMBL1498906

CCS(=O)(=O)c1ccc(-c2ccc(CC(C#N)NC(=O)[C@@H]3CCCCN3)cc2)c(C)c1

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSC P53634 20/20 0.63
CTSK P43235 5/20 0.63
KCNH2 Q12809 2/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2072993 1.00 CTSC (0.63) CTSCCTSKKCNH2
SCHEMBL4398633 1.00 CTSC (0.63) CTSCCTSKKCNH2
Trifluoroacetic Acid SCHEMBL2294609 0.95 CTSC (0.60) CTSCCTSKKCNH2
SCHEMBL3689681 0.90 CTSC (0.75) CTSCCTSKKCNH2
SCHEMBL3689684 0.90 CTSC (0.75) CTSCCTSKKCNH2
SCHEMBL2074014 0.87 CTSC (0.68) CTSCCTSKKCNH2
SCHEMBL2074012 0.87 CTSC (0.68) CTSCCTSKKCNH2
SCHEMBL1498932 0.84 CTSC (0.78) CTSCCTSKKCNH2
SCHEMBL2072316 0.83 CTSC (0.76) CTSCCTSKKCNH2
SCHEMBL2072318 0.83 CTSC (0.76) CTSCCTSKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2011506421-A 2011-03-03 JP claimed
EP-2231597-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS AstraZeneca AB (SE) 2010-09-29 EP claimed
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO claimed