SCHEMBL1499028

SCHEMBL1499028

N#Cc1ccc(-c2ccc([C@@H](C#N)CNC(=O)[C@@H]3CCCCN3)cc2)cc1F

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSC P53634 17/20 0.52
CTSK P43235 6/20 0.52
KCNH2 Q12809 2/20 0.52
EGLN2 Q96KS0 2/20 0.40
HTR2C P28335 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1499101 0.85 CTSC (0.51) CTSCCTSKKCNH2HTR2C
SCHEMBL1499181 0.85 CTSC (0.61) CTSCCTSKKCNH2HTR2C
SCHEMBL1498990 0.84 CTSC (0.52) CTSCCTSKKCNH2HTR2C
SCHEMBL1499071 0.83 CTSC (0.49) CTSCCTSKKCNH2HTR2C
SCHEMBL2075023 0.81 CTSC (0.76) CTSCCTSKKCNH2
SCHEMBL1499026 0.81 CTSC (0.76) CTSCCTSKKCNH2
SCHEMBL3657635 0.81 CTSC (0.60) CTSCCTSKKCNH2HTR2C
SCHEMBL1499171 0.80 CTSC (0.50) CTSCCTSKKCNH2HTR2C
SCHEMBL4247301 0.80 CTSC (0.49) CTSCCTSKKCNH2HTR2C
SCHEMBL4247298 0.80 CTSC (0.49) CTSCCTSKKCNH2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2011506421-A 2011-03-03 JP claimed
EP-2231597-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS AstraZeneca AB (SE) 2010-09-29 EP claimed
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO claimed