SCHEMBL15018564

SCHEMBL15018564

CC(C)(C)CCCCCC(=O)OOC(C)(C)c1ccccc1.CC(O)CC(C)(C)OOC(=O)CCCCCC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.35
NAAA Q02083 1/20 0.31
KCNH2 Q12809 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31
ADRB3 P13945 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ALOX15 P16050 1/20 0.31
HDAC3 O15379 2/20 0.30
HDAC4 P56524 2/20 0.30
HDAC1 Q13547 2/20 0.30
HDAC7 Q8WUI4 2/20 0.30
HDAC2 Q92769 2/20 0.30
HDAC10 Q969S8 2/20 0.30
HDAC11 Q96DB2 2/20 0.30
HDAC8 Q9BY41 2/20 0.30
HDAC6 Q9UBN7 2/20 0.30
HDAC9 Q9UKV0 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL216989 0.88 MAPK1 (0.44) MAPK1KCNH2CYP3A4CYP2C9ALDH1A1
SCHEMBL10714649 0.86 MAPT (0.37) LMNA
SCHEMBL215144 0.86 MAPT (0.37) LMNA
SCHEMBL30672047 0.85 MAPK1 (0.37) MAPK1NAAAKCNH2CYP3A4CYP2C9
SCHEMBL29253653 0.83 MAPT (0.34) ALDH1A1ALOX15HDAC11LMNA
SCHEMBL5184632 0.82 MAPK1 (0.43) MAPK1KCNH2CYP3A4CYP2C9ALDH1A1
SCHEMBL9863530 0.82 CNR1 (0.37) MAPK1CYP3A4ALDH1A1HDAC3HDAC4
SCHEMBL439547 0.81 MAPT (0.36) LMNA
SCHEMBL9616935 0.80 CNR1 (0.34) MAPK1KCNH2CYP3A4CYP2C9HDAC3
SCHEMBL11228688 0.79 CYP2D6 (0.37) CYP2C9HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10117974-B2 Non-fouling, anti-microbial, anti-thrombogenic graft-from compositions ARROW INTERNATIONAL, INC. (US) 2018-11-06 US disclosed
EP-2790746-B1 SURFACE MODIFICATION FOR CATHETERS COMPRISED OF MULTIPLE MATERIALS ARROW INT INC (US) 2018-05-09 EP disclosed
US-9895469-B2 Articles having non-fouling surfaces and processes for preparing the same including applying a primer coat ARROW INTERNATIONAL, INC. (US) 2018-02-20 US disclosed
US-9795762-B2 Surface modification for dialysis catheters ARROW INTERNATIONAL, INC. (US) 2017-10-24 US disclosed
EP-2790745-B1 LUMINAL MODIFICATIONS FOR CATHETERS ARROW INT INC (US) 2017-09-27 EP disclosed
US-9764069-B2 Articles having non-fouling surfaces and processes for preparing the same including pretreatment of articles SEMPRUS BIOSCIENCES CORPORATION (US) 2017-09-19 US disclosed
US-9694114-B2 Antimicrobial catheters with permeabilization agents ARROW INTERNATIONAL, INC. (US) 2017-07-04 US disclosed
US-20160235893-A1 ANTIMICROBIAL CATHETERS WITH PERMEABILIZATION AGENTS JPMORGAN CHASE BANK, N.A., AS ADMINISTRATIVE AGENT 2016-08-18 US disclosed
US-20160146974-A1 REDOX PROCESSES FOR CONTACT LENS MODIFICATION TELEFLEX LIFE SCIENCES LIMITED (MT) 2016-05-26 US disclosed
US-9120119-B2 Redox processes for contact lens modification SEMPRUS BIOSCIENCES CORPORATION (US) 2015-09-01 US disclosed
WO-2013090813-A1 REDOX PROCESSES FOR CONTACT LENS MODIFICATION SEMPRUS BIOSCIENCES CORP. (US) 2013-06-20 WO disclosed
US-20130155370-A1 SURFACE MODIFIED CONTACT LENSES SEMPRUS BIOSCIENCES CORP. (US) 2013-06-20 US disclosed
US-20130158211-A1 IMBIBING PROCESS FOR CONTACT LENS SURFACE MODIFICATION SEMPRUS BIOSCIENCES CORP. (US) 2013-06-20 US disclosed
WO-2013090801-A1 MULTISTEP UV PROCESS TO CREATE SURFACE MODIFIED CONTACT LENSES SEMPRUS BIOSCIENCES CORP. (US) 2013-06-20 WO disclosed
US-20130158150-A1 MULTISTEP UV PROCESS TO CREATE SURFACE MODIFIED CONTACT LENSES SEMPRUS BIOSCIENCES CORP. (US) 2013-06-20 US disclosed
US-20130155371-A1 REDOX PROCESSES FOR CONTACT LENS MODIFICATION SEMPRUS BIOSCIENCES CORP. (US) 2013-06-20 US disclosed
WO-2013090808-A1 HIGH IONIC STRENGTH PROCESS FOR CONTACT LENS MODIFICATION SEMPRUS BIOSCIENCES CORP. (US) 2013-06-20 WO disclosed
US-20130158517-A1 SURFACE MODIFICATION FOR DIALYSIS CATHETERS SEMPRUS BIOSCIENCES CORP. (US) 2013-06-20 US disclosed
WO-2013090780-A1 SURFACE MODIFIED CONTACT LENSES SEMPRUS BIOSCIENCES CORP. (US) 2013-06-20 WO disclosed
US-20130158518-A1 SURFACE MODIFICATION FOR CATHETERS COMPRISED OF MULTIPLE MATERIALS SEMPRUS BIOSCIENCES CORP. (US) 2013-06-20 US disclosed