SCHEMBL15038313

SCHEMBL15038313

COC(=O)c1cnc(N)nc1C(F)(F)F

nearest known ligand 0.72

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.72
MAPT P10636 3/20 0.53
GAA P10253 2/20 0.50
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 1/20 0.47
NFKB1 P19838 5/20 0.46
ATF1 P18846 2/20 0.46
CFTR P13569 2/20 0.46
JUN P05412 3/20 0.43
NFKB2 Q00653 3/20 0.43
RELA Q04206 3/20 0.43
LMNA P02545 1/20 0.43
PKM P14618 1/20 0.43
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12775325 0.86 KDM4E (0.54) KDM4EMAPTGAAALDH1A1CFTR
SCHEMBL3922065 0.84 KDM4E (1.00) KDM4EMAPTALDH1A1KMT2ANFKB1
SCHEMBL4592101 0.83 MAPT (0.57) KDM4EMAPTGAAALDH1A1KMT2A
SCHEMBL6475927 0.82 MAPT (0.60) KDM4EMAPTGAAALDH1A1KMT2A
Water SCHEMBL4593114 0.81 MAPT (0.56) KDM4EMAPTGAAALDH1A1KMT2A
SCHEMBL473934 0.81 ATF1 (0.62) KDM4EMAPTGAAALDH1A1KMT2A
SCHEMBL1759818 0.81 MAPT (0.53) KDM4EMAPTGAAALDH1A1KMT2A
SCHEMBL4888133 0.80 KDM4E (0.61) KDM4EALDH1A1KMT2ANFKB1ATF1
SCHEMBL29038495 0.78 TSHR (0.47) KDM4EMAPTGAAALDH1A1NFKB1
SCHEMBL30468126 0.78 TSHR (0.47) KDM4EMAPTGAAALDH1A1NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318389-B1 PYRIDAZINE DERIVATIVES AS SMO INHIBITORS NOVARTIS AG (CH) 2013-06-19 EP disclosed