SCHEMBL15049569

SCHEMBL15049569

COC(=O)c1cn(Cc2ccc(OC)cc2)nc1C(F)(F)F

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.59
KLKB1 P03952 17/20 0.55
DGAT1 O75907 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1049941 0.90 GAA (0.56) GAAKLKB1DGAT1
SCHEMBL2361709 0.89 GAA (0.54) GAAKLKB1DGAT1
SCHEMBL3355699 0.89 GAA (0.54) GAAKLKB1DGAT1
SCHEMBL7980023 0.88 KLKB1 (0.60) GAAKLKB1DGAT1
SCHEMBL20521837 0.88 GAA (0.53) GAAKLKB1DGAT1
SCHEMBL3356363 0.86 GAA (0.51) GAAKLKB1DGAT1
SCHEMBL14150628 0.83 KLKB1 (0.48) GAAKLKB1DGAT1
SCHEMBL1048741 0.83 KLKB1 (0.48) GAAKLKB1DGAT1
SCHEMBL371016 0.82 KMT2A (0.46) GAA
SCHEMBL14823853 0.82 KMT2A (0.46) GAAKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2456769-B1 NOVEL PYRAZOLE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX PHARMA SA (CH) 2013-06-26 EP disclosed