SCHEMBL15049635

SCHEMBL15049635

N#Cc1sc(Oc2cccc(Cl)n2)nc1-c1cn[nH]c1.N#Cc1sc(Oc2ccccn2)nc1-c1cn[nH]c1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 2/20 0.37
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
KCNH2 Q12809 1/20 0.32
CDC7 O00311 1/20 0.32
DBF4 Q9UBU7 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ILK Q13418 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1047866 0.93 CYP11B1 (0.36) GRM4CYP11B1CYP11B2CDC7DBF4
SCHEMBL1051493 0.92 GRM4 (0.42) GRM4KCNH2CDC7DBF4KDM4E
SCHEMBL1000214 0.80 GRM4 (0.45) GRM4KCNH2KDM4EILK
SCHEMBL366105 0.70 GRM4 (0.70) GRM4KCNH2
SCHEMBL1051726 0.67 CYP11B1 (0.41) CYP11B1CYP11B2
SCHEMBL1049256 0.66 GRM4 (0.57) GRM4KCNH2KDM4EILK
SCHEMBL13306656 0.61 GRM4 (0.41) GRM4CDC7DBF4KDM4EILK
SCHEMBL15049877 0.61 GRM4 (0.48) GRM4KCNH2KDM4EILK
SCHEMBL3288656 0.60 CNR2 (0.47) GRM4KCNH2
SCHEMBL22783773 0.59 PIK3CD (0.43) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2456769-B1 NOVEL PYRAZOLE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX PHARMA SA (CH) 2013-06-26 EP claimed