SCHEMBL15054832

SCHEMBL15054832

COc1c(N2CC[C@@H](CCNC(C)=O)C2)c(F)cc2c(=O)c3c(O)c(C(C)=O)sc3n(C3CC3)c12

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.47
TOP1 P11387 6/20 0.40
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 3/20 0.39
HPGD P15428 2/20 0.39
POLB P06746 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
PRKD3 O94806 1/20 0.39
ALOX15 P16050 1/20 0.39
OPRM1 P35372 1/20 0.39
CLK2 P49760 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
LMNA P02545 2/20 0.38
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15054591 0.95 KCNH2 (0.48) KCNH2TOP1KDM4EALDH1A1HPGD
SCHEMBL15053742 0.93 KCNH2 (0.48) KCNH2TOP1KDM4EALDH1A1HPGD
SCHEMBL15053743 0.93 KCNH2 (0.48) KCNH2TOP1KDM4EALDH1A1HPGD
SCHEMBL537045 0.89 KCNH2 (0.59) KCNH2TOP1
SCHEMBL15052748 0.89 KCNH2 (0.59) KCNH2TOP1
SCHEMBL15052745 0.89 KCNH2 (0.59) KCNH2TOP1
SCHEMBL15053067 0.88 KCNH2 (0.49) KCNH2TOP1KDM4EALDH1A1HPGD
SCHEMBL15053071 0.88 KCNH2 (0.49) KCNH2TOP1KDM4EALDH1A1HPGD
SCHEMBL15077891 0.86 KCNH2 (0.44) KCNH2TOP1KDM4EALDH1A1HPGD
SCHEMBL15052961 0.86 KCNH2 (0.42) KCNH2TOP1KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013096785-A1 2-SUBSTITUTED-THIENOQUINOLONES AND RELATED COMPOUNDS AS ANTI-INFECTIVE AGENTS ACHILLION PHARMACEUTICALS, INC. (US) 2013-06-27 WO claimed