SCHEMBL15060068

SCHEMBL15060068

CCn1nc(-c2cnccn2)cc1-c1cnc2[nH]c(-c3cnccc3C)cc2c1.Cc1cc(S(C)(=O)=O)ncc1-c1cnc2[nH]c(-c3cnccc3C)cc2c1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.34
ORAI1 Q96D31 1/20 0.32
CLK2 P49760 1/20 0.31
CLK3 P49761 1/20 0.31
DYRK1A Q13627 1/20 0.31
GCK P35557 1/20 0.31
PTGS2 P35354 1/20 0.30
MAP4K1 Q92918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15020844 0.89 HTR2C (0.34) KITCLK2CLK3DYRK1A
SCHEMBL15021244 0.84 ORAI1 (0.41) ORAI1CLK2CLK3DYRK1APTGS2
SCHEMBL15020834 0.82 PIK3C3 (0.35) KITORAI1
SCHEMBL15036344 0.80 CLK2 (0.38) KITCLK2CLK3DYRK1A
SCHEMBL12745918 0.77 CLK2 (0.39) CLK2CLK3DYRK1A
SCHEMBL15020511 0.77 ORAI1 (0.41) KITORAI1CLK2DYRK1APTGS2
SCHEMBL15020532 0.76 CYP17A1 (0.45) KITORAI1PTGS2
SCHEMBL15020476 0.76 BRD4 (0.43) KIT
SCHEMBL15020878 0.73 CYP19A1 (0.40) KITCLK2CLK3DYRK1A
SCHEMBL1460211 0.71 CLK2 (0.47) KITCLK2CLK3DYRK1APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013092467-A1 7-AZAINDOLE INHIBITORS OF CRAC F. HOFFMANN-LA ROCHE AG (CH) 2013-06-27 WO claimed