SCHEMBL15062313

SCHEMBL15062313

CC1(C)Oc2cc(N)ccc2C(c2ccc(Cl)cn2)=C1C#N

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
BACE1 P56817 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C19 P33261 2/20 0.32
KDM4E B2RXH2 2/20 0.32
MAPT P10636 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C9 P11712 1/20 0.31
PTGES O14684 1/20 0.31
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14670353 0.81 CYP3A4 (0.32) GRM5BACE1CYP3A4CYP2C19CYP2C9
SCHEMBL3023334 0.80 NR3C2 (0.38) BACE1
SCHEMBL13431070 0.76 BACE1 (0.31) BACE1
SCHEMBL15062302 0.75 GRM5 (0.34) GRM5BACE1CYP1A2
SCHEMBL3025613 0.74 MAPT (0.38) MEN1KMT2AKDM4EMAPTHPGD
SCHEMBL12085058 0.70 BACE1 (0.34) GRM5BACE1
SCHEMBL15062301 0.70
SCHEMBL14670455 0.70 BACE1 (0.35) GRM5BACE1
SCHEMBL3017342 0.69 KDM4E (0.39) MEN1KMT2ACYP3A4CYP2C19KDM4E
SCHEMBL3011515 0.69 NR3C2 (0.46) BACE1CYP3A4CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2179994-B1 FUSED BICYCLIC COMPOUND MITSUBISHI TANABE PHARMA CORP (JP) 2013-06-26 EP disclosed