SCHEMBL15062969

SCHEMBL15062969

CNC(=O)c1ccccc1-c1ccc2c(n1)CN(C(C)=O)c1cc(Cl)ccc1C=C2

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 14/20 0.53
NOTUM Q6P988 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
CGAS Q8N884 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15062968 1.00 HSD17B3 (0.53) HSD17B3NOTUML3MBTL1CGASKDM4E
SCHEMBL15063092 0.93 HSD17B3 (0.55) HSD17B3NOTUML3MBTL1
SCHEMBL15063091 0.93 HSD17B3 (0.55) HSD17B3NOTUML3MBTL1
SCHEMBL15062912 0.90 HSD17B3 (0.50) HSD17B3NOTUMKDM4E
SCHEMBL15062911 0.90 HSD17B3 (0.50) HSD17B3NOTUMKDM4E
SCHEMBL5046141 0.89 HSD17B3 (0.43) HSD17B3NOTUML3MBTL1CGASKDM4E
SCHEMBL5046143 0.89 HSD17B3 (0.43) HSD17B3NOTUML3MBTL1CGASKDM4E
SCHEMBL4803471 0.83 HSD17B3 (0.69) HSD17B3
SCHEMBL4803463 0.83 HSD17B3 (0.69) HSD17B3
SCHEMBL15063058 0.83 HSD17B3 (0.56) HSD17B3NOTUMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1725565-B1 FUSED HETEROTRICYCLIC COMPOUNDS AS INHIBITORS OF 17B-HYDROXYSTEROID DEHYDROGENASE 3 BRISTOL MYERS SQUIBB CO (US) 2013-07-03 EP disclosed