SCHEMBL15067429

SCHEMBL15067429

CC(=O)c1ccc(Nc2nccc3c(Nc4ccsc4)c(C)ccc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 13/20 0.56
RAF1 P04049 8/20 0.56
CSF1R P07333 4/20 0.56
DDR1 Q08345 4/20 0.56
DDR2 Q16832 4/20 0.56
TTBK1 Q5TCY1 1/20 0.41
TTBK2 Q6IQ55 1/20 0.41
LCK P06239 5/20 0.41
TEK Q02763 5/20 0.41
KDR P35968 3/20 0.39
TDO2 P48775 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
NPC1 O15118 4/20 0.37
RAB9A P51151 3/20 0.37
TDP1 Q9NUW8 2/20 0.37
MAPK14 Q16539 1/20 0.35
USP2 O75604 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15068724 0.88 BRAF (0.45) BRAFRAF1CSF1RDDR1DDR2
SCHEMBL15069205 0.87 BRAF (0.44) BRAFRAF1CSF1RDDR1DDR2
SCHEMBL15068707 0.84 BRAF (0.55) BRAFRAF1CSF1RDDR1DDR2
SCHEMBL15069790 0.84 BRAF (0.43) BRAFRAF1CSF1RDDR1DDR2
SCHEMBL15069219 0.84 BRAF (0.44) BRAFRAF1CSF1RDDR1DDR2
SCHEMBL15067507 0.82 BRAF (0.55) BRAFRAF1CSF1RDDR1DDR2
SCHEMBL27985926 0.82 BRAF (0.47) BRAFRAF1CSF1RDDR1DDR2
SCHEMBL15069773 0.80 BRAF (0.46) BRAFRAF1CSF1RDDR1DDR2
SCHEMBL27985938 0.80 BRAF (0.42) BRAFRAF1CSF1RDDR1DDR2
SCHEMBL15069808 0.80 BRAF (0.43) BRAFRAF1CSF1RDDR1DDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104039798-A Thieno[3,2-d]pyrimidine derivatives having inhibitory activity for protein kinases HANMI PHARM IND CO LTD 2014-09-10 CN claimed
EP-2797927-A1 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY FOR PROTEIN KINASES Hanmi Pharm. Co., Ltd. (KR) 2014-11-05 EP disclosed
CN-104039798-A Thieno[3,2-d]pyrimidine derivatives having inhibitory activity for protein kinases HANMI PHARM IND CO LTD 2014-09-10 CN disclosed
WO-2013100632-A1 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY FOR PROTEIN KINASES HANMI PHARM CO., LTD. (KR) 2013-07-04 WO disclosed