SCHEMBL15069293

SCHEMBL15069293

Cn1cc(-c2cc(N)ccc2Oc2ccc(F)cc2F)c2cc[nH]c2c1=O

nearest known ligand 0.76

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 20/20 0.76
BRD2 P25440 1/20 0.68
ADORA2B P29275 1/20 0.68
TSPO P30536 1/20 0.68
EP300 Q09472 1/20 0.68
BRD3 Q15059 1/20 0.68
BRDT Q58F21 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15771094 0.90 BRD4 (0.71) BRD4
SCHEMBL15069351 0.90 BRD4 (0.70) BRD4
SCHEMBL23436760 0.89 BRD4 (0.77) BRD4BRD2ADORA2BTSPOEP300
SCHEMBL15069650 0.89 BRD4 (0.81) BRD4
SCHEMBL23436641 0.89 BRD4 (0.76) BRD4BRD2ADORA2BTSPOEP300
SCHEMBL21652764 0.88 BRD4 (0.65) BRD4
SCHEMBL20384384 0.87 BRD4 (0.78) BRD4BRD2ADORA2BTSPOEP300
SCHEMBL31073856 0.87 BRD4 (0.72) BRD4BRD2ADORA2BTSPOEP300
SCHEMBL20384227 0.87 BRD4 (0.74) BRD4BRD2ADORA2BTSPOEP300
SCHEMBL21652831 0.86 BRD4 (0.68) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119684283-A Pyrrolo [2,3-c ] pyridines and use thereof 山东新时代药业有限公司 2025-03-25 CN disclosed
WO-2024193527-A1 PYRROLO[2,3-C]PYRIDINE COMPOUND AS BROMODOMAIN INHIBITOR 山东新时代药业有限公司 2024-09-26 WO disclosed
WO-2024054955-A1 HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. (US) 2024-03-14 WO disclosed
WO-2024054955-A1 HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE HALDA THERAPEUTICS OPCO, INC. (US) 2024-03-14 WO disclosed
US-20230158039-A1 BROMODOMAIN INHIBITORS ABBVIE INC (US) 2023-05-25 US disclosed
CN-109384785-B Pyrrolopyridinone derivatives, preparation method and medical application thereof 浙江海正药业股份有限公司 2021-09-28 CN disclosed
US-20210236508-A1 BROMODOMAIN INHIBITORS ABBVIE INC (US) 2021-08-05 US disclosed
EP-3828183-A1 SULFOXIMINE COMPOUND AS BROMODOMAIN PROTEIN INHIBITOR AND PHARMACEUTICAL COMPOSITION AND MEDICAL USE THEREOF Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2021-06-02 EP disclosed
CN-106986872-B Bromodomain inhibitors 艾伯维公司 2020-04-21 CN disclosed
WO-2020020288-A1 SULFOXIMINE COMPOUND AS BROMODOMAIN PROTEIN INHIBITOR AND PHARMACEUTICAL COMPOSITION AND MEDICAL USE THEREOF 正大天晴药业集团股份有限公司 2020-01-30 WO disclosed
WO-2020007322-A1 COMPOUND TARGETED TO DEGRADE BET PROTEIN AND APPLICATION THEREOF 清华大学 2020-01-09 WO disclosed
US-20180296566-A1 BROMODOMAIN INHIBITORS ABBVIE INC (US) 2018-10-18 US disclosed
EP-2797918-B1 BROMODOMAIN INHIBITORS ABBVIE INC (US) 2017-11-29 EP disclosed
US-20160143916-A1 BROMODOMAIN INHIBITORS ABBVIE INC (US) 2016-05-26 US disclosed
US-9296741-B2 Bromodomain inhibitors ABBVIE INC. (US) 2016-03-29 US disclosed
EP-2797918-A1 BROMODOMAIN INHIBITORS AbbVie Inc. (US) 2014-11-05 EP disclosed
US-20140162971-A1 BROMODOMAIN INHIBITORS ABBVIE INC. 2014-06-12 US disclosed
WO-2013097601-A1 BROMODOMAIN INHIBITORS ABBVIE INC. (US) 2013-07-04 WO disclosed
WO-2013097052-A1 BROMODOMAIN INHIBITORS ABBOTT LABORATORIES (US) 2013-07-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180296566-A1 BROMODOMAIN INHIBITORS BRD4, BRD1, BRD3 BRD4 1/4885BRD2 4/4885ADORA2B 832/4885
US-20140162971-A1 BROMODOMAIN INHIBITORS BRD4, BRD1, BRD3 BRD4 1/4885BRD2 4/4885ADORA2B 832/4885
US-20230158039-A1 BROMODOMAIN INHIBITORS BRD4, BRD1, BRD3 BRD4 1/4885BRD2 4/4885ADORA2B 832/4885
US-20160143916-A1 BROMODOMAIN INHIBITORS BRD4, BRD1, BRD3 BRD4 1/4885BRD2 4/4885ADORA2B 832/4885
US-20210236508-A1 BROMODOMAIN INHIBITORS BRD4, BRD1, BRD3 BRD4 1/4885BRD2 4/4885ADORA2B 832/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.