SCHEMBL15072073

SCHEMBL15072073

Cc1cnc(Nc2cnn(CC(F)F)c2)nc1N(N)C[C@H]1CCN(CCC#N)C1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 13/20 0.43
JAK3 P52333 12/20 0.43
JAK1 P23458 11/20 0.43
STAT3 P40763 9/20 0.43
TYK2 P29597 9/20 0.43
ABL1 P00519 3/20 0.42
KDR P35968 3/20 0.42
GSK3B P49841 3/20 0.42
AURKB Q96GD4 3/20 0.42
TBK1 Q9UHD2 3/20 0.36
IKBKE Q14164 1/20 0.36
BTK Q06187 1/20 0.36
FLT3 P36888 1/20 0.36
MAP3K14 Q99558 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15059532 0.84 JAK2 (0.45) JAK2JAK3JAK1STAT3TYK2
SCHEMBL15059530 0.84 JAK2 (0.45) JAK2JAK3JAK1STAT3TYK2
SCHEMBL2582400 0.74 JAK3 (0.43) JAK2JAK3JAK1STAT3TYK2
SCHEMBL16337534 0.71 JAK3 (0.45) JAK2JAK3JAK1STAT3TYK2
SCHEMBL16336319 0.71 JAK3 (0.45) JAK2JAK3JAK1STAT3TYK2
SCHEMBL15059211 0.71 JAK3 (0.43) JAK2JAK3JAK1AURKBBTK
SCHEMBL15059213 0.71 JAK3 (0.43) JAK2JAK3JAK1AURKBBTK
SCHEMBL15058843 0.71 JAK3 (0.45) JAK2JAK3JAK1TBK1BTK
SCHEMBL15058844 0.71 JAK3 (0.45) JAK2JAK3JAK1TBK1BTK
SCHEMBL15060038 0.70 JAK1 (0.45) JAK2JAK3JAK1STAT3TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013092854-A1 PYRIMIDINE-2,4-DIAMINE DERIVATIVES AS KINASE INHIBITORS CELLZOME LIMITED (GB) 2013-06-27 WO disclosed