SCHEMBL15077709

SCHEMBL15077709

CN(c1ncnc2[nH]ccc12)C1CC2CCNCC2C1

nearest known ligand 0.66

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 19/20 0.66
JAK3 P52333 10/20 0.66
JAK2 O60674 9/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16234625 1.00 JAK1 (0.66) JAK1JAK3JAK2
SCHEMBL15077702 1.00 JAK1 (0.66) JAK1JAK3JAK2
SCHEMBL16199578 1.00 JAK1 (0.66) JAK1JAK3JAK2
SCHEMBL15077581 1.00 JAK1 (0.66) JAK1JAK3JAK2
Hydrochloric Acid SCHEMBL18493482 0.99 JAK1 (0.65) JAK1JAK3JAK2
Hydrochloric Acid SCHEMBL16192278 0.99 JAK1 (0.65) JAK1JAK3JAK2
Hydrochloric Acid SCHEMBL16192276 0.99 JAK1 (0.65) JAK1JAK3JAK2
SCHEMBL15077726 0.93 JAK1 (0.62) JAK1JAK3JAK2
Hydrochloric Acid SCHEMBL18493460 0.92 JAK1 (0.61) JAK1JAK3JAK2
Hydrochloric Acid SCHEMBL16192313 0.92 JAK1 (0.61) JAK1JAK3JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2796460-B1 PYRROLE SIX-MEMBERED HETEROARYL RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND MEDICINAL USES THEREOF JIANGSU HENGRUI MEDICINE CO (CN) 2018-07-04 EP disclosed
WO-2013091539-A1 PYRROLE SIX-MEMBERED HETEROARYL RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND MEDICINAL USES THEREOF 江苏恒瑞医药股份有限公司 (CN) 2013-06-27 WO disclosed