SCHEMBL15080867

SCHEMBL15080867

Cc1ccc(NCCNc2nc(-c3ccc(Cl)cc3Cl)cn3nc(CN4CCN(C)CC4)cc23)nc1N

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 0.52
GSK3A P49840 1/20 0.40
FGFR1 P11362 1/20 0.34
KDR P35968 1/20 0.34
LMNA P02545 1/20 0.34
CRHR1 P34998 4/20 0.33
CCNT1 O60563 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ALPL P05186 1/20 0.32
HRH4 Q9H3N8 2/20 0.32
HTR3A P46098 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12835855 0.83 GSK3B (0.74) GSK3BGSK3AFGFR1CCNT1HRH4
SCHEMBL8131726 0.82 GSK3B (0.64) GSK3BGSK3ALMNACCNT1
SCHEMBL12835876 0.81 GSK3B (0.53) GSK3BGSK3AALDH1A1
SCHEMBL8143251 0.78 GSK3B (0.45) GSK3BGSK3AKDM4EALDH1A1ALPL
SCHEMBL1514117 0.78 POLB (0.43) GSK3BLMNAKDM4EALDH1A1POLB
Trifluoroacetic Acid SCHEMBL1514015 0.76 GSK3B (0.45) GSK3BGSK3AKDM4EALDH1A1
SCHEMBL8145934 0.75 GSK3B (0.69) GSK3BGSK3A
SCHEMBL8135071 0.74 GSK3B (0.73) GSK3BGSK3ACCNT1
SCHEMBL12835842 0.74 GSK3B (0.72) GSK3BGSK3ALMNACCNT1KDM4E
Hydrochloric Acid SCHEMBL1514127 0.73 GSK3B (0.71) GSK3BGSK3AFGFR1LMNACCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8476267-B2 Imidazo-, pyrazolopyrazines and imidazotriazines and their use BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-07-02 US disclosed