SCHEMBL15085658

SCHEMBL15085658

COc1cc2c(Nc3ccc(Cl)c(Cl)c3)ncnc2cc1OCc1nc(N2CCN(C(C)(C)C)CC2)no1

nearest known ligand 0.84

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EPHA2 P29317 19/20 0.84
EPHB4 P54760 14/20 0.84
KDR P35968 16/20 0.84
ERBB2 P04626 3/20 0.82
EGFR P00533 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL906808 0.91 EPHA2 (1.00) EPHA2EPHB4KDRERBB2EGFR
Hydrochloric Acid SCHEMBL907153 0.91 EPHA2 (0.98) EPHA2EPHB4KDRERBB2EGFR
SCHEMBL906935 0.90 EPHA2 (1.00) EPHA2EPHB4KDRERBB2EGFR
SCHEMBL907272 0.90 EPHA2 (1.00) EPHA2EPHB4KDRERBB2EGFR
Hydrochloric Acid SCHEMBL907249 0.89 EPHA2 (0.98) EPHA2EPHB4KDRERBB2EGFR
SCHEMBL907073 0.89 EPHA2 (1.00) EPHA2EPHB4KDRERBB2EGFR
Hydrochloric Acid SCHEMBL910764 0.88 EPHA2 (0.98) EPHA2EPHB4KDRERBB2EGFR
SCHEMBL906934 0.88 EPHA2 (1.00) EPHA2EPHB4KDRERBB2EGFR
SCHEMBL13590284 0.84 EPHA2 (0.90) EPHA2EPHB4KDRERBB2
SCHEMBL3031854 0.81 EPHA2 (0.85) EPHA2EPHB4KDRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8481001-B2 Combination therapies comprising quinoxaline inhibitors of P13K-alpha for use in the treatment of cancer EXELIXIS, INC. (US) 2013-07-09 US disclosed