SCHEMBL1509481

SCHEMBL1509481

CN1CCCC2(CCCN(CCc3ccc(NC(=O)c4ccc5[nH]c(-c6cc(-c7cccnc7O)ccc6O)nc5c4)cc3)C2)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.39
ABCG2 Q9UNQ0 2/20 0.39
ADORA2A P29274 1/20 0.37
CLK2 P49760 1/20 0.37
CLK3 P49761 1/20 0.37
DYRK1A Q13627 1/20 0.37
DDR2 Q16832 1/20 0.36
HPSE Q9Y251 8/20 0.35
POLB P06746 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
PRSS12 P56730 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14090392 0.95 HDAC6 (0.40) ABCB1ABCG2ADORA2ACLK2CLK3
SCHEMBL12834518 0.91 ABCB1 (0.39) ABCB1ABCG2ADORA2ACLK2CLK3
SCHEMBL14090393 0.88 ABCG2 (0.43) ABCB1ABCG2ADORA2AHPSEHDAC3
SCHEMBL1509560 0.86 ABCG2 (0.41) ABCB1ABCG2ADORA2AHPSEHDAC3
SCHEMBL12833673 0.84 ABCB1 (0.43) ABCB1ABCG2ADORA2AHPSEHDAC3
SCHEMBL1509459 0.84 ABCG2 (0.42) ABCB1ABCG2ADORA2AHPSEHDAC3
SCHEMBL12833553 0.83 HDAC6 (0.50) ABCB1ABCG2ADORA2ADDR2HPSE
SCHEMBL14090449 0.80 ABCG2 (0.44) ABCB1ABCG2ADORA2AHPSE
SCHEMBL14090399 0.79 KIT (0.43) ABCB1ABCG2ADORA2ADDR2HPSE
SCHEMBL14531512 0.79 ABCG2 (0.39) ABCB1ABCG2ADORA2ADDR2HPSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298770-A1 Heterocyclic compounds as TrkA modulators ChemBridge Corporation (US) 2011-03-23 EP disclosed