SCHEMBL15095355

SCHEMBL15095355

CN[C@@H](C)C(=O)N[C@H](C(=O)N1CC[C@H]2NC[C@H](C(=O)Nc3cccc4ccccc34)[C@H]21)C(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
XIAP P98170 15/20 0.49
CASP9 P55211 1/20 0.41
CYP3A4 P08684 3/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 1/20 0.39
KDM4E B2RXH2 1/20 0.39
BIRC2 Q13490 5/20 0.38
BIRC3 Q13489 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2632208 0.85 XIAP (0.49) XIAPCASP9CYP3A4CYP2C9CYP2C19
SCHEMBL2117250 0.85 XIAP (0.49) XIAPCASP9CYP3A4CYP2C9CYP2C19
SCHEMBL2115163 0.84 XIAP (0.42) XIAPCYP3A4CYP2C9CYP2C19KDM4E
SCHEMBL2632124 0.83 XIAP (0.48) XIAPCASP9CYP3A4CYP2C9CYP2C19
SCHEMBL2113168 0.82 XIAP (0.46) XIAPCASP9CYP3A4CYP2C9CYP2C19
SCHEMBL2632123 0.82 XIAP (0.46) XIAPCASP9CYP3A4CYP2C9CYP2C19
SCHEMBL23847519 0.81 XIAP (0.45) XIAPCASP9CYP3A4CYP2C9KDM4E
SCHEMBL2631846 0.81 XIAP (0.45) XIAPCASP9CYP3A4CYP2C9KDM4E
SCHEMBL13048262 0.81 XIAP (0.45) XIAPCASP9CYP3A4CYP2C9KDM4E
SCHEMBL2113161 0.81 XIAP (0.45) XIAPCASP9CYP3A4CYP2C9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8481495-B2 IAP inhibitors TETRALOGIC PHARMACEUTICALS CORPORATION (US) 2013-07-09 US disclosed