SCHEMBL1509665

SCHEMBL1509665

COc1cccc2c1CCc1cnc(-n3ncc(C(=O)Nc4ccc(CCN5CCN(C)CC5)cc4)c3N)nc1-2

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 18/20 0.45
ABCG2 Q9UNQ0 17/20 0.45
SCN5A Q14524 1/20 0.42
SCN9A Q15858 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C8 P10632 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
ABCC1 P33527 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4757948 0.79 NPC1 (0.45) SCN5ASCN9A
SCHEMBL14090024 0.73 ABCG2 (0.40) ABCB1ABCG2CYP1A2CYP2C8CYP2D6
SCHEMBL14090004 0.73 IKBKB (0.42) ABCB1ABCG2CYP1A2CYP2C8CYP2D6
SCHEMBL14091169 0.72 EGFR (0.44) ABCB1ABCG2CYP1A2CYP2C8CYP2D6
SCHEMBL14091172 0.71 FLT3 (0.39) ABCB1ABCG2
SCHEMBL14090162 0.71 IKBKB (0.40) ABCB1ABCG2CYP1A2CYP2C8CYP2D6
SCHEMBL14090038 0.70 CSF1R (0.38) ABCB1ABCG2CYP1A2CYP2C8CYP2D6
SCHEMBL14090045 0.70 FLT3 (0.40) ABCB1ABCG2
SCHEMBL14090047 0.69 CSF1R (0.40) ABCB1ABCG2
SCHEMBL14089982 0.69 MAPT (0.42) SCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298770-A1 Heterocyclic compounds as TrkA modulators ChemBridge Corporation (US) 2011-03-23 EP disclosed