SCHEMBL15212654

SCHEMBL15212654

COc1ccc(CCN)cc1-c1ccnc2cc(-c3cc(OC)c(OC)c(OC)c3)oc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4C Q08493 2/20 0.41
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
KDM4E B2RXH2 1/20 0.40
ATM Q13315 1/20 0.40
CYP1A2 P05177 2/20 0.38
TSHR P16473 2/20 0.38
CYP3A4 P08684 1/20 0.38
NFKB1 P19838 1/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1B1 Q16678 1/20 0.38
BRD4 O60885 2/20 0.38
ADORA2A P29274 1/20 0.38
LMNA P02545 2/20 0.38
MEN1 O00255 1/20 0.38
APEX1 P27695 1/20 0.38
KMT2A Q03164 1/20 0.38
TAAR1 Q96RJ0 2/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15210548 0.88 PDE4C (0.37) PDE4CHTR2AHTR2CHTR2BKDM4E
SCHEMBL723374 0.85 PDE4C (0.39) PDE4CCYP1A2CYP1A1CYP1B1BRD4
SCHEMBL721309 0.83 PDE4C (0.47) PDE4CCYP1A2CYP1A1CYP1B1BRD4
SCHEMBL723398 0.82 CALCRL (0.50) PDE4CCYP1A2CYP3A4CYP1A1CYP1B1
SCHEMBL723093 0.81 PDE4C (0.55) PDE4CKDM4ECYP1A2CYP3A4CYP1A1
SCHEMBL15210399 0.81 KDM4E (0.48) PDE4CHTR2AHTR2CHTR2BKDM4E
SCHEMBL16429216 0.80 PDE4C (0.40) PDE4CKDM4ECYP1A2CYP3A4CYP1A1
SCHEMBL15210645 0.80 PDE4C (0.40) PDE4CKDM4ECYP1A2CYP3A4CYP1A1
SCHEMBL723977 0.80 CFTR (0.42) KDM4EBRD4LMNAMEN1KMT2A
SCHEMBL725317 0.80 FYN (0.45) PDE4CCYP1A2CYP3A4CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817313-A1 FUROPYRIDINE DERIVATIVES Merck Patent GmbH (DE) 2014-12-31 EP disclosed
WO-2013124025-A1 FUROPYRIDINE DERIVATIVES MERCK PATENT GMBH (DE) 2013-08-29 WO disclosed