SCHEMBL15214151

SCHEMBL15214151

Cc1ccc([C@H](C)n2cc(C#N)cc(C(=O)c3ccc(-n4cnc(C)c4)c(C)c3)c2=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
HTT P42858 1/20 0.43
PSEN1 P49768 10/20 0.37
PSEN2 P49810 10/20 0.37
APH1B Q8WW43 10/20 0.37
NCSTN Q92542 10/20 0.37
APH1A Q96BI3 10/20 0.37
PSENEN Q9NZ42 10/20 0.37
LDLR P01130 1/20 0.37
PCSK9 Q8NBP7 1/20 0.37
USP30 Q70CQ3 1/20 0.33
BRD4 O60885 2/20 0.33
SIGMAR1 Q99720 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
USP2 O75604 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12712780 0.93 PSEN1 (0.45) ALDH1A1HTTPSEN1PSEN2APH1B
SCHEMBL15214141 0.85 PSEN1 (0.47) ALDH1A1HTTPSEN1PSEN2APH1B
SCHEMBL15214173 0.84 BRD4 (0.37) ALDH1A1HTTPSEN1PSEN2APH1B
SCHEMBL8077510 0.84 PSEN1 (0.57) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL15214154 0.83 PSEN1 (0.39) ALDH1A1HTTPSEN1PSEN2APH1B
SCHEMBL12712793 0.80 PSEN1 (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL12712823 0.79 PSEN1 (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL15214149 0.78 PSEN1 (0.39) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL12712867 0.78 PSEN1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL12712828 0.78 PSEN1 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8518975-B2 Gamma secretase modulators Merck Sharp + Dohme Corp. (US) 2013-08-27 US disclosed