SCHEMBL15214839

SCHEMBL15214839

N#Cc1c(-c2ccc(I)cc2)c[nH]c1N

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GRM5 P41594 1/20 0.33
ADORA2A P29274 5/20 0.32
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 3/20 0.32
HPGD P15428 2/20 0.32
PPARG P37231 1/20 0.32
STAT3 P40763 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
NR2E3 Q9Y5X4 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
ADORA1 P30542 6/20 0.32
HSD17B10 Q99714 2/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
NTRK1 P04629 2/20 0.31
PIK3CA P42336 1/20 0.31
DYRK1A Q13627 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27423329 0.83 ADORA1 (0.46) MEN1KMT2AADORA2AKDM4EALDH1A1
SCHEMBL1905542 0.83 ADORA1 (0.46) NPSR1MEN1KMT2AADORA2AKDM4E
SCHEMBL3783457 0.83 KDM4E (0.48) NPSR1MEN1KMT2AADORA2AKDM4E
SCHEMBL6236169 0.82 ADORA1 (0.47) NPSR1MEN1KMT2AGRM5ADORA2A
SCHEMBL18269174 0.79 ADORA1 (0.35) NPSR1MEN1KMT2AGRM5ADORA2A
SCHEMBL22283897 0.79 ADORA1 (0.51) NPSR1MEN1KMT2AADORA2AKDM4E
SCHEMBL10226576 0.79 CYP2A6 (0.42) NPSR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL4482253 0.76 IKBKB (0.47) MEN1KMT2AALDH1A1HPGDMAPT
SCHEMBL2618362 0.76 MEN1 (0.44) NPSR1MEN1KMT2AGRM5ADORA2A
SCHEMBL7026138 0.72 AS3MT (0.54) MAPTPIM1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8518970-B2 Compounds and methods of use ABBVIE INC. (US) 2013-08-27 US disclosed