SCHEMBL15215848

SCHEMBL15215848

CNc1nccc(-c2cccnc2Oc2cc(C(=O)O)ccc2C)n1

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.68
TEK Q02763 13/20 0.68
YES1 P07947 1/20 0.67
AURKB Q96GD4 11/20 0.62
AURKA O14965 9/20 0.61
TPX2 Q9ULW0 6/20 0.61
LCK P06239 4/20 0.55
ABL1 P00519 1/20 0.55
CSF1R P07333 1/20 0.55
KIT P10721 1/20 0.55
SRC P12931 1/20 0.55
MAPK14 Q16539 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1265373 0.91 KDR (0.69) KDRTEKYES1AURKBAURKA
SCHEMBL1265588 0.88 KDR (0.80) KDRTEKYES1AURKBAURKA
SCHEMBL2296344 0.88 TEK (0.66) KDRTEKYES1AURKBAURKA
SCHEMBL1265555 0.86 KDR (0.61) KDRTEKYES1AURKBAURKA
SCHEMBL1264019 0.86 KDR (0.66) KDRTEKYES1AURKBAURKA
SCHEMBL1264824 0.86 KDR (0.66) KDRTEKYES1AURKBAURKA
SCHEMBL1264726 0.85 KDR (0.72) KDRTEKYES1AURKBAURKA
SCHEMBL1265978 0.85 KDR (0.72) KDRTEKYES1AURKBAURKA
SCHEMBL5312489 0.85 KDR (0.62) KDRTEKYES1AURKBAURKA
SCHEMBL1265135 0.84 KDR (0.64) KDRTEKYES1AURKBAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130226549-A1 STRUCTURE-BASED FRAGMENT HOPPING FOR LEAD OPTIMIZATION AND IMPROVEMENT IN SYNTHETIC ACCESSIBILITY TSENG, YUFENG J. (TW) 2013-08-29 US disclosed