SCHEMBL1521673

SCHEMBL1521673

CNc1cc2c(cn1)CN(c1cc(NC(=O)NC(C)c3cccnc3)c(F)cc1C)C(=O)N2C

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 10/20 0.38
NAMPT P43490 3/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP2C9 P11712 2/20 0.35
TNK2 Q07912 3/20 0.34
MAP4K2 Q12851 3/20 0.34
BMX P51813 2/20 0.34
TRPV1 Q8NER1 1/20 0.33
CHRM4 P08173 1/20 0.33
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33
RIPK1 Q13546 1/20 0.33
RIPK3 Q9Y572 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1521655 0.93 MAPK1 (0.41) MAPK1
SCHEMBL1521984 0.93 MAPK1 (0.41) MAPK1
SCHEMBL1521653 0.93 MAPK1 (0.41) MAPK1
SCHEMBL1521647 0.87 RAF1 (0.37) TNK2MAP4K2BMXABL1
SCHEMBL1521797 0.80 TNK2 (0.37) TNK2MAP4K2BMXTRPV1ABL1
SCHEMBL1521766 0.79 TNK2 (0.42) TNK2MAP4K2BMXABL1BCR
SCHEMBL1521979 0.77 RAF1 (0.37) TNK2MAP4K2BMXABL1BCR
SCHEMBL1521678 0.77 KDR (0.40) TNK2MAP4K2BMXABL1BCR
SCHEMBL1521554 0.77 BRAF (0.48)
SCHEMBL1521960 0.77 BRAF (0.37) TNK2MAP4K2BMXABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7897762-B2 Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS, LLC (US) 2011-03-01 US claimed
US-20090099190-A1 Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS, LLC (US) 2009-04-16 US claimed
US-20110118271-A1 Kinase Inhibitors Useful For The Treatment Of Proliferative Diseases FLYNN DANIEL L 2011-05-19 US disclosed
US-7897762-B2 Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS, LLC (US) 2011-03-01 US disclosed
US-20090099190-A1 Kinase inhibitors useful for the treatment of proliferative diseases DECIPHERA PHARMACEUTICALS, LLC (US) 2009-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110118271-A1 Kinase Inhibitors Useful For The Treatment Of Proliferative Diseases BRAF, PRKDC, RAF1 MAPK1 93/4885NAMPT 661/4885KMT2A 1762/4885
US-20090099190-A1 Kinase inhibitors useful for the treatment of proliferative diseases BRAF, PRKDC, RAF1 MAPK1 93/4885NAMPT 661/4885KMT2A 1762/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.