SCHEMBL15310563

SCHEMBL15310563

CC(N)(CCCc1ccc(Sc2cccc(C(F)(F)F)c2)cc1F)COP(=O)(O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 14/20 0.47
S1PR3 Q99500 7/20 0.45
S1PR5 Q9H228 3/20 0.39
S1PR4 O95977 2/20 0.39
SIRT2 Q8IXJ6 1/20 0.36
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 1/20 0.35
HPGD P15428 2/20 0.35
MEN1 O00255 1/20 0.35
S1PR2 O95136 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
ALOX12 P18054 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TLR9 Q9NR96 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11949089 1.00 S1PR1 (0.47) S1PR1S1PR3S1PR5S1PR4SIRT2
SCHEMBL11888754 0.90 S1PR1 (0.54) S1PR1S1PR3S1PR5S1PR4SIRT2
SCHEMBL11888753 0.90 S1PR1 (0.54) S1PR1S1PR3S1PR5S1PR4SIRT2
SCHEMBL4339103 0.87 S1PR1 (0.37) S1PR1S1PR3SIRT2SLC6A2SLC6A4
SCHEMBL4339109 0.87 S1PR1 (0.37) S1PR1S1PR3SIRT2SLC6A2SLC6A4
SCHEMBL11888760 0.85 S1PR1 (0.56) S1PR1S1PR3S1PR5S1PR4SIRT2
SCHEMBL11888761 0.85 S1PR1 (0.56) S1PR1S1PR3S1PR5S1PR4SIRT2
SCHEMBL4339107 0.85 SLC6A2 (0.36) S1PR1S1PR3SIRT2SLC6A2SLC6A4
SCHEMBL3300524 0.84 SLC6A2 (0.40) S1PR1S1PR3SIRT2SLC6A2SLC6A4
SCHEMBL3300531 0.84 SLC6A2 (0.40) S1PR1S1PR3SIRT2SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058317-B1 AMINOPHOSPHORIC ACID ESTER DERIVATIVE AND S1P RECEPTOR MODULATOR CONTAINING THE SAME AS ACTIVE INGREDIENT KYORIN SEIYAKU KK (JP) 2013-10-16 EP disclosed