SCHEMBL15329602

SCHEMBL15329602

Cc1cccc2c(C=O)c(-c3ccc(F)c(F)c3F)[nH]c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRIM24 O15164 1/20 0.38
TRIM33 Q9UPN9 1/20 0.38
PDE7A Q13946 1/20 0.37
AHR P35869 1/20 0.36
KDM4E B2RXH2 3/20 0.36
CCNB2 O95067 1/20 0.36
CDK1 P06493 1/20 0.36
CCNB1 P14635 1/20 0.36
GSK3B P49841 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
CCNB3 Q8WWL7 1/20 0.36
KIF11 P52732 1/20 0.36
MAPT P10636 3/20 0.34
KMT2A Q03164 2/20 0.34
ATM Q13315 1/20 0.34
GAA P10253 2/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2554134 0.91 PDE7A (0.40) TRIM24TRIM33PDE7AAHRKDM4E
SCHEMBL15329563 0.88 FEN1 (0.36) GSK3BCDK5CDK5R1ALDH1A1MAPK10
SCHEMBL15331095 0.84 CCNB2 (0.42) TRIM24TRIM33PDE7AAHRKDM4E
SCHEMBL15332224 0.83 PARP1 (0.39) TRIM24TRIM33PDE7AAHRKDM4E
SCHEMBL15332951 0.83 PARP1 (0.39) TRIM24TRIM33PDE7AAHRKDM4E
SCHEMBL15329708 0.83 KDM4E (0.40) TRIM24TRIM33PDE7AAHRKDM4E
SCHEMBL15331976 0.82 CCNB2 (0.47) TRIM24TRIM33AHRKDM4ECCNB2
SCHEMBL2550909 0.81 TNKS (0.37) CCNB2CDK1CCNB1GSK3BCDK5
SCHEMBL2562309 0.81 PDE7A (0.43) TRIM24TRIM33PDE7AAHRKDM4E
SCHEMBL15329887 0.80 TNKS (0.38) TRIM24TRIM33PDE7AKDM4ECCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
US-20120126690-A1 ORGANIC ELECTROLUMINESCENCE DEVICE FUJIFILM CORPORATION 2012-05-24 US disclosed