SCHEMBL15329812

SCHEMBL15329812

COc1ccc(C(=O)NC(=O)Nc2ccc3c(c2)C(=Cc2ccc[nH]2)C(=O)N3)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 7/20 1.00
AURKB Q96GD4 9/20 0.87
KIT P10721 1/20 0.71
FLT4 P35916 1/20 0.71
KDR P35968 1/20 0.71
TLK2 Q86UE8 4/20 0.67
JAK3 P52333 1/20 0.67
PDPK1 O15530 4/20 0.65
PDGFRB P09619 1/20 0.64
NTRK1 P04629 1/20 0.62
AKT2 P31751 1/20 0.62
PDK1 Q15118 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15329805 1.00 FLT3 (1.00) FLT3AURKBKITFLT4KDR
SCHEMBL15328345 0.93 AURKB (1.00) FLT3AURKBKITFLT4KDR
SCHEMBL15328352 0.93 AURKB (1.00) FLT3AURKBKITFLT4KDR
SCHEMBL15328123 0.86 AURKB (1.00) FLT3AURKBKITFLT4KDR
SCHEMBL15328125 0.86 AURKB (1.00) FLT3AURKBKITFLT4KDR
SCHEMBL15327950 0.85 AURKB (0.74) FLT3AURKBKITFLT4KDR
SCHEMBL15327947 0.85 AURKB (0.74) FLT3AURKBKITFLT4KDR
SCHEMBL15328214 0.83 AURKB (1.00) FLT3AURKBKITFLT4KDR
SCHEMBL15327881 0.83 FLT3 (1.00) FLT3AURKBKITFLT4KDR
SCHEMBL15328216 0.83 AURKB (1.00) FLT3AURKBKITFLT4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2838531-B1 INDOLIN-2-ONE DERIVATIVES AS PROTEIN KINASE INHIBITORS ANNJI PHARM CO LTD (CN) 2016-09-21 EP claimed
US-20130281451-A1 INDOLIN-2-ONE DERIVATIVES AS PROTEIN KINASE INHIBITORS Annji Pharmaceutical Co., Ltd. (TW) 2013-10-24 US claimed
EP-2838531-B1 INDOLIN-2-ONE DERIVATIVES AS PROTEIN KINASE INHIBITORS ANNJI PHARM CO LTD (CN) 2016-09-21 EP disclosed
US-8946282-B2 Indolin-2-one derivatives as protein kinase inhibitors Annji Pharmaceutical Co., Ltd. (TW) 2015-02-03 US disclosed
US-20130281451-A1 INDOLIN-2-ONE DERIVATIVES AS PROTEIN KINASE INHIBITORS Annji Pharmaceutical Co., Ltd. (TW) 2013-10-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130281451-A1 INDOLIN-2-ONE DERIVATIVES AS PROTEIN KINASE INHIBITORS ING2, CDK2, MAP3K20 FLT3 1086/4885AURKB 100/4885KIT 1529/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.