SCHEMBL15397604

SCHEMBL15397604

CC(=O)N1CCC(C(=O)N2CC(NC(=O)Nc3ccc(Cl)cc3)C(c3ccc(Cl)c(Cl)c3)C2)CC1

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 0.67
TACR3 P29371 2/20 0.67
FPR1 P21462 6/20 0.59
FPR2 P25090 4/20 0.59
TACR2 P21452 13/20 0.58
TAC3 Q9UHF0 6/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15397605 1.00 TACR1 (0.67) TACR1TACR3FPR1FPR2TACR2
SCHEMBL13801644 0.87 TACR1 (0.65) TACR1TACR3TACR2TAC3
SCHEMBL4153912 0.87 TACR1 (0.65) TACR1TACR3TACR2TAC3
SCHEMBL4153915 0.87 TACR1 (0.65) TACR1TACR3TACR2TAC3
SCHEMBL12517759 0.83 TACR1 (0.59) TACR1TACR3TACR2TAC3
SCHEMBL13814682 0.81 TACR1 (0.67) TACR1TACR3TACR2TAC3
SCHEMBL4158529 0.81 TACR1 (0.67) TACR1TACR3TACR2TAC3
SCHEMBL13801638 0.81 TACR1 (0.67) TACR1TACR3TACR2TAC3
SCHEMBL4158533 0.81 TACR1 (0.67) TACR1TACR3TACR2TAC3
SCHEMBL4144164 0.81 TACR1 (0.67) TACR1TACR3TACR2TAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE49686-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-10 US disclosed
US-RE48334-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2020-12-01 US disclosed
US-8592454-B2 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-11-26 US disclosed