SCHEMBL15399178

SCHEMBL15399178

Cc1cc(C(C)(C)Cl)nc(N)n1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.62
HSP90AB1 P08238 3/20 0.62
NUDT1 P36639 2/20 0.44
HSD17B10 Q99714 1/20 0.40
MAPT P10636 1/20 0.40
CYP1A2 P05177 2/20 0.39
NPC1 O15118 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
CRHBP P24387 2/20 0.38
CRHR2 Q13324 2/20 0.38
TSHR P16473 1/20 0.38
CYP2D6 P10635 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
ATM Q13315 1/20 0.36
GRM4 Q14833 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15429553 0.83 HSP90AA1 (0.67) HSP90AA1HSP90AB1NUDT1HSD17B10MAPT
SCHEMBL5367782 0.82 HSP90AA1 (0.71) HSP90AA1HSP90AB1NUDT1HSD17B10MAPT
SCHEMBL27029868 0.77 KMT2A (0.45) HSP90AA1HSP90AB1MAPTNPC1RAB9A
SCHEMBL5361699 0.77 HSP90AA1 (1.00) HSP90AA1HSP90AB1NUDT1HSD17B10CYP1A2
SCHEMBL27269562 0.75 HSP90AA1 (0.34) HSP90AA1HSP90AB1
SCHEMBL151114 0.74
Ammonia Solution, Strong SCHEMBL20919221 0.71 HSP90AA1 (0.56) HSP90AA1HSP90AB1NUDT1MAPTCYP1A2
SCHEMBL30863954 0.71 HSP90AA1 (0.56) HSP90AA1HSP90AB1NUDT1MAPTCYP1A2
SCHEMBL27651209 0.71 HSP90AA1 (0.56) HSP90AA1HSP90AB1NUDT1MAPTCYP1A2
SCHEMBL150686 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140005172-A1 Benzoxazepines as Inhibitors of PI3K/M TOR and Methods of Their Use and Manufacture ELELIXIS, INC. (US) 2014-01-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140005172-A1 Benzoxazepines as Inhibitors of PI3K/M TOR and Methods of Their Use and Manufacture MTOR, RICTOR, PIK3R2 HSP90AA1 1580/4885HSP90AB1 829/4885NUDT1 3805/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.