SCHEMBL15418671

SCHEMBL15418671

NC1=N[C@]2(CCO1)c1cc(-c3cccnc3F)ccc1Oc1c(F)cc(N3CCC(F)(F)CC3)cc12

nearest known ligand 0.75

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.75
KCNH2 Q12809 4/20 0.67
CTSD P07339 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2522359 1.00 BACE1 (0.75) BACE1KCNH2CTSD
SCHEMBL15418855 0.93 BACE1 (0.87) BACE1KCNH2CTSD
SCHEMBL2371855 0.93 BACE1 (0.87) BACE1KCNH2CTSD
SCHEMBL15467552 0.93 BACE1 (0.87) BACE1KCNH2CTSD
SCHEMBL15418987 0.89 BACE1 (0.86) BACE1KCNH2CTSD
SCHEMBL2516520 0.89 BACE1 (0.86) BACE1KCNH2CTSD
SCHEMBL2522768 0.86 BACE1 (0.64) BACE1KCNH2CTSD
SCHEMBL2517624 0.86 BACE1 (0.64) BACE1KCNH2CTSD
SCHEMBL2524552 0.86 BACE1 (1.00) BACE1KCNH2CTSD
SCHEMBL2522310 0.86 BACE1 (1.00) BACE1KCNH2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547686-B1 AMINO-DIHYDROOXAZINE AND AMINO-DIHYDROTHIAZINE SPIRO COMPOUNDS AS BETA-SECRETASE MODULATORS AND THEIR MEDICAL USE AMGEN INC (US) 2014-01-22 EP disclosed