SCHEMBL15418752

SCHEMBL15418752

NC1=N[C@@]2(COC1)c1cc(-c3cncnc3)ccc1Oc1c(F)cc(C3=CCCOC3)cc12

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.58
KCNH2 Q12809 2/20 0.47
CTSD P07339 5/20 0.46
CTSE P14091 1/20 0.46
BACE2 Q9Y5Z0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2521167 0.91 BACE1 (0.62) BACE1KCNH2CTSDCTSEBACE2
SCHEMBL2521170 0.91 BACE1 (0.62) BACE1KCNH2CTSDCTSEBACE2
SCHEMBL6845777 0.90 BACE1 (0.56) BACE1KCNH2CTSDCTSEBACE2
SCHEMBL2523512 0.87 BACE1 (0.59) BACE1KCNH2CTSDCTSEBACE2
SCHEMBL2523509 0.87 BACE1 (0.59) BACE1KCNH2CTSDCTSEBACE2
SCHEMBL2381100 0.87 BACE1 (0.62) BACE1KCNH2CTSDCTSEBACE2
SCHEMBL2381098 0.87 BACE1 (0.62) BACE1KCNH2CTSDCTSEBACE2
SCHEMBL2524132 0.84 BACE1 (0.83) BACE1KCNH2CTSDCTSEBACE2
SCHEMBL2523553 0.84 BACE1 (0.83) BACE1KCNH2CTSDCTSEBACE2
SCHEMBL2523382 0.81 BACE1 (0.52) BACE1KCNH2CTSDCTSEBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547686-B1 AMINO-DIHYDROOXAZINE AND AMINO-DIHYDROTHIAZINE SPIRO COMPOUNDS AS BETA-SECRETASE MODULATORS AND THEIR MEDICAL USE AMGEN INC (US) 2014-01-22 EP disclosed