SCHEMBL15418804

SCHEMBL15418804

NC1=N[C@]2(CCO1)c1cc(-c3cccnc3F)ccc1Oc1c2cc(-c2ccccc2)nc1F

nearest known ligand 0.84

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.84
CTSD P07339 2/20 0.65
CTSE P14091 1/20 0.65
BACE2 Q9Y5Z0 1/20 0.65
KCNH2 Q12809 3/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15418889 1.00 BACE1 (0.84) BACE1CTSDCTSEBACE2KCNH2
SCHEMBL15418733 0.94 BACE1 (0.83) BACE1CTSDCTSEBACE2KCNH2
SCHEMBL15418781 0.94 BACE1 (0.83) BACE1CTSDCTSEBACE2KCNH2
SCHEMBL2526329 0.93 BACE1 (0.85) BACE1CTSDCTSEBACE2KCNH2
SCHEMBL2526327 0.93 BACE1 (0.85) BACE1CTSDCTSEBACE2KCNH2
SCHEMBL15418880 0.93 BACE1 (0.85) BACE1CTSDCTSEBACE2KCNH2
SCHEMBL2521392 0.91 BACE1 (1.00) BACE1CTSDCTSEBACE2KCNH2
SCHEMBL2521398 0.91 BACE1 (1.00) BACE1CTSDCTSEBACE2KCNH2
SCHEMBL15418704 0.91 BACE1 (0.85) BACE1CTSDCTSEBACE2
SCHEMBL2522589 0.91 BACE1 (0.85) BACE1CTSDCTSEBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547686-B1 AMINO-DIHYDROOXAZINE AND AMINO-DIHYDROTHIAZINE SPIRO COMPOUNDS AS BETA-SECRETASE MODULATORS AND THEIR MEDICAL USE AMGEN INC (US) 2014-01-22 EP disclosed