SCHEMBL15418873

SCHEMBL15418873

NC1=N[C@@]2(COC1)c1cc(-c3cc(F)ccc3F)ccc1Oc1ncc(C3CCOCC3)cc12

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.61
CTSD P07339 3/20 0.44
KCNH2 Q12809 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12213335 0.86 BACE1 (0.81) BACE1CTSDKCNH2
SCHEMBL15418814 0.86 BACE1 (0.50) BACE1CTSDKCNH2
SCHEMBL1994452 0.83 BACE1 (0.76) BACE1CTSDKCNH2
SCHEMBL15418883 0.83 BACE1 (0.62) BACE1CTSDKCNH2
SCHEMBL1994454 0.83 BACE1 (0.76) BACE1CTSDKCNH2
SCHEMBL2524963 0.83 BACE1 (0.60) BACE1CTSDKCNH2
SCHEMBL2524959 0.83 BACE1 (0.60) BACE1CTSDKCNH2
SCHEMBL15418856 0.82 BACE1 (0.50) BACE1CTSDKCNH2
SCHEMBL15418615 0.77 BACE1 (0.61) BACE1CTSDKCNH2
SCHEMBL15509615 0.76 BACE1 (1.00) BACE1CTSDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547686-B1 AMINO-DIHYDROOXAZINE AND AMINO-DIHYDROTHIAZINE SPIRO COMPOUNDS AS BETA-SECRETASE MODULATORS AND THEIR MEDICAL USE AMGEN INC (US) 2014-01-22 EP disclosed