SCHEMBL15418945

SCHEMBL15418945

NC1=NC2(CCO1)c1cc(-c3cccnc3)ccc1Oc1cnc(-c3cccnc3)cc12

nearest known ligand 0.66

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.66
CTSD P07339 9/20 0.66
KCNH2 Q12809 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15418634 0.92 BACE1 (0.64) BACE1CTSDKCNH2
SCHEMBL1995831 0.90 BACE1 (0.79) BACE1CTSDKCNH2
SCHEMBL15510061 0.90 BACE1 (0.79) BACE1CTSDKCNH2
SCHEMBL1995833 0.90 BACE1 (0.79) BACE1CTSDKCNH2
SCHEMBL15418743 0.89 BACE1 (0.84) BACE1CTSD
SCHEMBL15418688 0.89 BACE1 (0.84) BACE1CTSD
SCHEMBL15418970 0.88 BACE1 (0.64) BACE1CTSDKCNH2
SCHEMBL15418915 0.83 BACE1 (0.67) BACE1CTSDKCNH2
SCHEMBL15509448 0.82 BACE1 (0.71) BACE1CTSDKCNH2
SCHEMBL14878048 0.82 BACE1 (0.71) BACE1CTSDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547686-B1 AMINO-DIHYDROOXAZINE AND AMINO-DIHYDROTHIAZINE SPIRO COMPOUNDS AS BETA-SECRETASE MODULATORS AND THEIR MEDICAL USE AMGEN INC (US) 2014-01-22 EP disclosed