SCHEMBL15419418

SCHEMBL15419418

O=C(O)CNC(=O)c1c(O)n(C2CCOC(=O)C2)c(=O)n(C2CCCCC2)c1=O

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 14/20 0.78
EGLN2 Q96KS0 3/20 0.78
HIF1AN Q9NWT6 2/20 0.78
EGLN3 Q9H6Z9 2/20 0.78
OGFOD1 Q8N543 1/20 0.78
NPSR1 Q6W5P4 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
XBP1 P17861 2/20 0.45
MAPK1 P28482 2/20 0.45
MAPT P10636 1/20 0.45
ATM Q13315 1/20 0.45
BBOX1 O75936 1/20 0.37
ASPH Q12797 1/20 0.37
KDM8 Q8N371 1/20 0.37
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
USP2 O75604 1/20 0.32
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3424056 0.88 EGLN1 (0.86) EGLN1EGLN2HIF1ANEGLN3OGFOD1
SCHEMBL3422096 0.88 EGLN1 (1.00) EGLN1EGLN2HIF1ANEGLN3OGFOD1
SCHEMBL3422098 0.88 EGLN1 (1.00) EGLN1EGLN2HIF1ANEGLN3OGFOD1
SCHEMBL3421361 0.88 EGLN1 (1.00) EGLN1EGLN2HIF1ANEGLN3OGFOD1
SCHEMBL3423522 0.88 EGLN1 (1.00) EGLN1EGLN2HIF1ANEGLN3OGFOD1
SCHEMBL3419112 0.88 EGLN1 (1.00) EGLN1EGLN2HIF1ANEGLN3OGFOD1
SCHEMBL3423425 0.87 EGLN1 (0.97) EGLN1EGLN2HIF1ANEGLN3OGFOD1
SCHEMBL3419140 0.87 EGLN1 (0.97) EGLN1EGLN2HIF1ANEGLN3OGFOD1
Bicarbonate SCHEMBL15419071 0.87 EGLN1 (0.97) EGLN1EGLN2HIF1ANEGLN3OGFOD1
SCHEMBL3421189 0.87 EGLN1 (0.97) EGLN1EGLN2HIF1ANEGLN3OGFOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2037922-B9 PROLYL HYDROXYLASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2017-08-23 EP claimed
EP-2037922-B1 PROLYL HYDROXYLASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-22 EP claimed