SCHEMBL15428702

SCHEMBL15428702

Cc1ccc(Nc2ncc3cnn(C[C@H]4CC[C@H](N(C)C(=O)O)CC4)c3n2)cc1S(N)(=O)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 13/20 0.41
CDK2 P24941 2/20 0.41
CDK9 P50750 1/20 0.41
AURKA O14965 13/20 0.40
JAK2 O60674 3/20 0.40
TYK2 P29597 3/20 0.40
AURKB Q96GD4 3/20 0.40
PLK4 O00444 2/20 0.40
MAP4K4 O95819 2/20 0.40
LCK P06239 2/20 0.40
FYN P06241 2/20 0.40
CSF1R P07333 2/20 0.40
LYN P07948 2/20 0.40
RET P07949 2/20 0.40
ROS1 P08922 2/20 0.40
KIT P10721 2/20 0.40
FGFR1 P11362 2/20 0.40
SRC P12931 2/20 0.40
FLT1 P17948 2/20 0.40
FGFR3 P22607 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL342943 0.91 CDK1 (0.39) CDK1CDK2CDK9AURKAJAK2
SCHEMBL342942 0.91 CDK1 (0.39) CDK1CDK2CDK9AURKAJAK2
SCHEMBL15428699 0.88 CDK1 (0.41) CDK1CDK2CDK9AURKAJAK2
SCHEMBL342956 0.88 CDK1 (0.39) CDK1CDK2CDK9AURKAJAK2
SCHEMBL15428718 0.87 CDK2 (0.47) CDK1CDK2CDK9AURKAJAK2
SCHEMBL344726 0.87 CDK1 (0.42) CDK1CDK2CDK9AURKAJAK2
SCHEMBL343043 0.87 MERTK (0.42) CDK1CDK2AURKAJAK2TYK2
SCHEMBL343868 0.87 CDK1 (0.41) CDK1CDK2CDK9AURKAJAK2
SCHEMBL343044 0.87 MERTK (0.42) CDK1CDK2AURKAJAK2TYK2
SCHEMBL10167396 0.87 CDK1 (0.41) CDK1CDK2CDK9AURKAJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8637529-B2 Pyrazolo[3,4-d]pyrimidine compounds AbbYie Inc. (US) 2014-01-28 US disclosed