SCHEMBL1543089

SCHEMBL1543089

COc1c(C(C)(C)C)cc(Br)cc1C(C)(CO)Cc1ccc(NS(C)(=O)=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
TRPV1 Q8NER1 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTPRB P23467 3/20 0.38
EPHX2 P34913 1/20 0.38
NR1H4 Q96RI1 1/20 0.38
PTPN2 P17706 1/20 0.36
PTPN1 P18031 1/20 0.36
PTPRA P18433 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1542804 0.89 CYP3A4 (0.44) CYP3A4TRPV1KDM4EALDH1A1LMNA
SCHEMBL1543087 0.83 CYP3A4 (0.44) CYP3A4TRPV1EPHX2NR1H4
SCHEMBL1542651 0.82 CYP3A4 (0.43) CYP3A4TRPV1KDM4EALDH1A1LMNA
SCHEMBL1542803 0.75 CYP3A4 (0.44) CYP3A4TRPV1EPHX2NR1H4
SCHEMBL1542505 0.74 CYP3A4 (0.47) CYP3A4LMNAHPGDSMN1; SMN2
SCHEMBL2128771 0.74 CYP3A4 (0.45) CYP3A4TRPV1EPHX2NR1H4
SCHEMBL6765973 0.73 CYP3A4 (0.62) CYP3A4ALDH1A1LMNASMN1; SMN2
SCHEMBL12678845 0.72 CYP3A4 (0.44) CYP3A4ALDH1A1LMNAHPGDHTT
SCHEMBL1542649 0.72 CYP3A4 (0.44) CYP3A4TRPV1EPHX2NR1H4
SCHEMBL1764621 0.72 CYP3A4 (0.46) CYP3A4TRPV1KDM4ELMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307372-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2011-04-13 EP disclosed
WO-2010010017-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-01-28 WO disclosed