SCHEMBL15436282

SCHEMBL15436282

C[C@H](Nc1nc(Nc2cnccn2)cc(N2CCC(OC(=O)O)CC2)n1)c1ccc(F)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 4/20 0.51
JAK3 P52333 3/20 0.51
JAK1 P23458 1/20 0.51
TYK2 P29597 1/20 0.51
KCNH2 Q12809 2/20 0.41
NTRK1 P04629 2/20 0.41
HRH3 Q9Y5N1 2/20 0.40
IDH1 O75874 3/20 0.39
CYP2C9 P11712 1/20 0.39
EPHX2 P34913 1/20 0.39
ACACB O00763 4/20 0.38
KDM4E B2RXH2 1/20 0.38
PRCP P42785 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1365720 0.90 JAK2 (0.52) JAK2JAK3JAK1TYK2KCNH2
SCHEMBL1365716 0.90 JAK2 (0.52) JAK2JAK3JAK1TYK2KCNH2
SCHEMBL1368051 0.89 JAK2 (0.48) JAK2JAK3JAK1TYK2NTRK1
SCHEMBL1368012 0.88 JAK2 (0.55) JAK2JAK3JAK1TYK2KCNH2
SCHEMBL1368007 0.88 JAK2 (0.55) JAK2JAK3JAK1TYK2KCNH2
SCHEMBL1368609 0.88 JAK2 (0.51) JAK2JAK3JAK1TYK2KCNH2
SCHEMBL1368605 0.88 JAK2 (0.51) JAK2JAK3JAK1TYK2KCNH2
Hydrochloric Acid SCHEMBL1368475 0.88 JAK2 (0.54) JAK2JAK3JAK1TYK2KCNH2
Hydrochloric Acid SCHEMBL1368478 0.88 JAK2 (0.54) JAK2JAK3JAK1TYK2KCNH2
Hydrochloric Acid SCHEMBL1368927 0.87 JAK2 (0.51) JAK2JAK3JAK1TYK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394999-B1 AMINOPYRAZINE DERIVATIVE AND MEDICINE NIPPON SHINYAKU CO LTD (JP) 2014-01-29 EP claimed