SCHEMBL15463520

SCHEMBL15463520

c1ccc(-c2ncn(C3CCN(Cc4ccon4)CC3)c2-c2ccncn2)cc1

nearest known ligand 0.63

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 5/20 0.63
CSNK1E P49674 5/20 0.63
MAPK14 Q16539 14/20 0.50
MAPK13 O15264 2/20 0.38
MAPK12 P53778 2/20 0.38
MAPK11 Q15759 2/20 0.38
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1639943 0.91 CSNK1D (0.77) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL1640957 0.86 CSNK1D (0.84) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL1640975 0.86 CSNK1D (0.69) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL1639876 0.84 MAPK14 (0.52) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL15203571 0.84 CSNK1D (0.64) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL1639785 0.79 CSNK1D (0.60) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL1640763 0.78 CSNK1D (0.59) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL1640309 0.78 CSNK1D (0.59) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL1640953 0.78 CSNK1D (1.00) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL1640205 0.77 CSNK1D (0.57) CSNK1DCSNK1EMAPK14MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493876-B1 IMIDAZOLE DERIVATIVES AS CASEIN KINASE INHIBITORS PFIZER (US) 2014-02-12 EP disclosed