SCHEMBL15463536

SCHEMBL15463536

CN(C(=O)C(F)(F)F)[C@@H]1CCN(C(=O)O)CC1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.56
TACR2 P21452 19/20 0.56
TAC3 Q9UHF0 6/20 0.56
TACR3 P29371 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4002700 1.00 TACR1 (0.56) TACR1TACR2TAC3TACR3
SCHEMBL4150577 1.00 TACR1 (0.56) TACR1TACR2TAC3TACR3
SCHEMBL30693203 0.87 TACR1 (0.52) TACR1TACR2TAC3TACR3
SCHEMBL1968592 0.87 TACR1 (0.52) TACR1TACR2TAC3TACR3
SCHEMBL4157210 0.86 TACR1 (0.75) TACR1TACR2TAC3TACR3
SCHEMBL4157211 0.86 TACR1 (0.75) TACR1TACR2TAC3TACR3
SCHEMBL4143844 0.84 TACR2 (0.78) TACR1TACR2TAC3TACR3
SCHEMBL4156962 0.84 TACR2 (0.78) TACR1TACR2TAC3TACR3
SCHEMBL4156957 0.84 TACR2 (0.78) TACR1TACR2TAC3TACR3
SCHEMBL4157907 0.84 TACR2 (0.78) TACR1TACR2TAC3TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2336105-B9 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL (JP) 2014-09-17 EP disclosed
EP-2336105-B1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL (JP) 2014-02-12 EP disclosed