SCHEMBL15463557

SCHEMBL15463557

CN(C(=O)N(C)[C@H]1CN(C(=O)O)C[C@H]1c1ccc(F)cc1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.73
TACR2 P21452 11/20 0.73
TACR3 P29371 12/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15397687 1.00 TACR1 (0.73) TACR1TACR2TACR3
SCHEMBL15397596 1.00 TACR1 (0.73) TACR1TACR2TACR3
SCHEMBL15397688 1.00 TACR1 (0.73) TACR1TACR2TACR3
SCHEMBL15397569 1.00 TACR1 (0.73) TACR1TACR2TACR3
SCHEMBL15397490 0.94 TACR1 (0.66) TACR1TACR2TACR3
SCHEMBL15397597 0.93 TACR1 (0.65) TACR1TACR2TACR3
SCHEMBL15397667 0.93 TACR1 (0.65) TACR1TACR2TACR3
SCHEMBL1971258 0.92 TACR1 (0.81) TACR1TACR2TACR3
SCHEMBL15397548 0.91 TACR1 (0.77) TACR1TACR2TACR3
SCHEMBL15397485 0.91 TACR1 (0.77) TACR1TACR2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2336105-B9 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL (JP) 2014-09-17 EP disclosed
EP-2336105-B1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL (JP) 2014-02-12 EP disclosed