SCHEMBL15510022

SCHEMBL15510022

COC(C)(C)C#Cc1cnc2c(c1)[C@@]1(COC(N)=N1)c1cc(-c3cccnc3)ccc1O2

nearest known ligand 0.77

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.77
BACE2 Q9Y5Z0 4/20 0.77
KCNH2 Q12809 10/20 0.71
CTSD P07339 2/20 0.55
CTSE P14091 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014606 1.00 BACE1 (0.77) BACE1BACE2KCNH2CTSDCTSE
SCHEMBL2012465 1.00 BACE1 (0.77) BACE1BACE2KCNH2CTSDCTSE
SCHEMBL2011246 0.94 BACE1 (0.70) BACE1BACE2KCNH2CTSD
SCHEMBL15509845 0.94 BACE1 (0.70) BACE1BACE2KCNH2CTSD
SCHEMBL15509866 0.94 BACE1 (0.70) BACE1BACE2KCNH2CTSD
SCHEMBL15509653 0.92 BACE1 (0.76) BACE1BACE2KCNH2CTSDCTSE
SCHEMBL2019582 0.92 BACE1 (0.76) BACE1BACE2KCNH2CTSDCTSE
SCHEMBL2013687 0.92 BACE1 (0.76) BACE1BACE2KCNH2CTSDCTSE
SCHEMBL2007830 0.92 BACE1 (0.84) BACE1BACE2KCNH2CTSDCTSE
SCHEMBL2007833 0.92 BACE1 (0.84) BACE1BACE2KCNH2CTSDCTSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2328903-B1 SPIRO-TETRACYCLIC RING COMPOUNDS AS BETASECRETASE MODULATORS AND METHODS OF USE AMGEN INC (US) 2014-03-05 EP disclosed