SCHEMBL15512697

SCHEMBL15512697

CC(=O)CCCCC[C@H](NC(=O)CCN1CCCCC1)c1ncc(-c2ccccc2)[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 20/20 1.00
HDAC2 Q92769 4/20 0.58
HDAC3 O15379 3/20 0.58
HDAC6 Q9UBN7 3/20 0.58
HDAC8 Q9BY41 1/20 0.58
HDAC4 P56524 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2072117 0.95 HDAC1 (0.90) HDAC1HDAC2HDAC3HDAC6HDAC8
SCHEMBL15512832 0.87 HDAC1 (1.00) HDAC1HDAC2HDAC3HDAC6HDAC8
SCHEMBL4416660 0.84 HDAC1 (0.72) HDAC1HDAC2HDAC3HDAC6HDAC8
SCHEMBL15512857 0.83 HDAC1 (1.00) HDAC1HDAC2HDAC3HDAC6HDAC8
Trifluoroacetic Acid SCHEMBL2071732 0.82 HDAC1 (0.91) HDAC1HDAC2HDAC3HDAC6HDAC8
SCHEMBL15513585 0.81 HDAC1 (1.00) HDAC1HDAC2HDAC3HDAC6HDAC8
SCHEMBL17183344 0.81 HDAC1 (0.69) HDAC1HDAC3
SCHEMBL15707523 0.81 HDAC1 (0.69) HDAC1HDAC3
SCHEMBL15514069 0.81 HDAC1 (1.00) HDAC1HDAC2HDAC3HDAC6HDAC8
SCHEMBL15513645 0.81 HDAC1 (1.00) HDAC1HDAC2HDAC3HDAC6HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828171-B1 HETEROCYCLE DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ANGELETTI P IST RICHERCHE BIO (IT) 2014-03-12 EP claimed