SCHEMBL15512966

SCHEMBL15512966

O=C(O)CCCCC[C@H](NC(=O)c1cncs1)c1ncc(-c2ccc3ccccc3c2)[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 16/20 1.00
HDAC3 O15379 17/20 0.84
HDAC2 Q92769 9/20 0.73
HDAC8 Q9BY41 4/20 0.73
KCNH2 Q12809 1/20 0.69
HDAC10 Q969S8 1/20 0.69
HDAC11 Q96DB2 1/20 0.69
HDAC6 Q9UBN7 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2073154 0.95 HDAC1 (0.91) HDAC1HDAC3HDAC2HDAC8KCNH2
SCHEMBL15513583 0.93 HDAC1 (0.86) HDAC1HDAC3HDAC2HDAC8KCNH2
SCHEMBL17183330 0.91 HDAC1 (1.00) HDAC1HDAC3HDAC2HDAC8
SCHEMBL5276057 0.91 HDAC1 (1.00) HDAC1HDAC3HDAC2HDAC8
SCHEMBL22501408 0.91 HDAC1 (0.83) HDAC1HDAC3HDAC2HDAC8KCNH2
SCHEMBL22501409 0.91 HDAC1 (0.83) HDAC1HDAC3HDAC2HDAC8KCNH2
SCHEMBL17145325 0.90 HDAC1 (0.81) HDAC1HDAC3HDAC2HDAC8KCNH2
SCHEMBL22501455 0.89 HDAC3 (0.81) HDAC1HDAC3HDAC2HDAC8KCNH2
Trifluoroacetic Acid SCHEMBL2071588 0.89 HDAC1 (0.80) HDAC1HDAC3HDAC2HDAC8KCNH2
Trifluoroacetic Acid SCHEMBL2071707 0.88 HDAC1 (0.90) HDAC1HDAC3HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828171-B1 HETEROCYCLE DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ANGELETTI P IST RICHERCHE BIO (IT) 2014-03-12 EP claimed
US-9150527-B2 Metalloenzyme inhibitor compounds INNOCRIN PHARMACEUTICALS, INC. (US) 2015-10-06 US disclosed