SCHEMBL15513797

SCHEMBL15513797

CCC(=O)CCCCC[C@H](NC(=O)C(=O)N1CCN(C)CC1)c1ncc(-c2cc(OC)c3ccccc3n2)[nH]1

nearest known ligand 0.81

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 19/20 0.81
HDAC3 O15379 11/20 0.54
HDAC6 Q9UBN7 11/20 0.54
HDAC2 Q92769 10/20 0.54
HDAC8 Q9BY41 10/20 0.54
KCNH2 Q12809 3/20 0.54
CYP2C9 P11712 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2073028 0.96 HDAC1 (0.76) HDAC1HDAC3HDAC6HDAC2HDAC8
SCHEMBL15513112 0.90 HDAC1 (1.00) HDAC1HDAC3HDAC6HDAC2HDAC8
Hydrochloric Acid SCHEMBL2071316 0.88 HDAC1 (0.90) HDAC1HDAC3HDAC6HDAC2HDAC8
SCHEMBL15513047 0.88 HDAC1 (1.00) HDAC1HDAC3HDAC6HDAC2HDAC8
Hydrochloric Acid SCHEMBL2070943 0.87 HDAC1 (0.99) HDAC1HDAC3HDAC6HDAC2HDAC8
SCHEMBL2074146 0.87 HDAC1 (0.83) HDAC1HDAC3HDAC6HDAC2HDAC8
SCHEMBL15512699 0.87 HDAC1 (1.00) HDAC1HDAC3HDAC6HDAC2HDAC8
Trifluoroacetic Acid SCHEMBL2074169 0.86 HDAC1 (0.92) HDAC1HDAC3HDAC6HDAC2HDAC8
Hydrochloric Acid SCHEMBL2073855 0.86 HDAC1 (0.99) HDAC1HDAC3HDAC6HDAC2HDAC8
SCHEMBL15518456 0.85 HDAC1 (0.79) HDAC1HDAC3HDAC6HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828171-B1 HETEROCYCLE DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ANGELETTI P IST RICHERCHE BIO (IT) 2014-03-12 EP claimed