SCHEMBL15519370

SCHEMBL15519370

CC1(C)CC(=O)Nc2c(Br)cccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 6/20 0.46
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
AHR P35869 2/20 0.35
PDK2 Q15119 3/20 0.34
PDK4 Q16654 2/20 0.34
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
PDK1 Q15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5764522 0.81 PDE7A (0.46) PDE7ACA12CA1CA2CA4
SCHEMBL17478594 0.79 PDE7A (0.45) PDE7ACA12CA1CA2CA4
SCHEMBL6221451 0.79 AHR (0.54) PDE7ACA12CA1CA2CA4
SCHEMBL10587563 0.79 TYMS (0.38) AHRPDK2PDK4RARBRARG
SCHEMBL6221081 0.78 PDK2 (0.58) AHRPDK2PDK4RARBRARG
SCHEMBL15135472 0.76 RARB (0.36) CA12CA1CA2CA4CA7
SCHEMBL3079489 0.76 PDK2 (0.44) AHRPDK2PDK4RARBRARG
SCHEMBL9378647 0.74 TDP1 (0.41) TSHR
SCHEMBL31117008 0.73 PDK2 (0.61) PDE7ACA12CA1CA2CA4
SCHEMBL17397785 0.73 PDE7A (0.39) PDE7ACA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2582667-B1 HETEROCYCLIC SUBSTITUTED METHOXYPHENYL DERIVATIVES WITH OXOGROUP, METHOD FOR PRODUCING SAME AND USE AS GPR40 RECEPTOR MODULATORS SANOFI SA (FR) 2014-03-19 EP disclosed