SCHEMBL15524465

SCHEMBL15524465

CC(C)(C)OC(=O)N(CCO)Cc1ccc(N)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.50
HDAC3 O15379 4/20 0.44
HDAC1 Q13547 4/20 0.44
HDAC2 Q92769 4/20 0.44
NCOR2 Q9Y618 3/20 0.44
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
MAPT P10636 1/20 0.36
CA14 Q9ULX7 1/20 0.36
ADRB3 P13945 1/20 0.36
USP2 O75604 2/20 0.35
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18067962 0.93 HDAC3 (0.46) SSTR4HDAC3HDAC1HDAC2NCOR2
SCHEMBL16682332 0.90 HDAC3 (0.51) SSTR4HDAC3HDAC1HDAC2NCOR2
SCHEMBL3141997 0.89 HDAC1 (0.49) SSTR4HDAC3HDAC1HDAC2NCOR2
SCHEMBL16682328 0.89 ADRB3 (0.44) SSTR4HDAC3HDAC1HDAC2NCOR2
SCHEMBL13767869 0.87 HDAC3 (0.43) SSTR4HDAC3HDAC1HDAC2NCOR2
SCHEMBL14002386 0.87 SSTR4 (0.51) SSTR4HDAC3HDAC1HDAC2NCOR2
SCHEMBL18067948 0.86 ADRB3 (0.42) SSTR4HDAC3HDAC1HDAC2NCOR2
SCHEMBL3142415 0.86 MAPT (0.51) HDAC3HDAC1HDAC2NCOR2MAPT
SCHEMBL2258889 0.86 SSTR4 (0.50) SSTR4HDAC3HDAC1HDAC2NCOR2
SCHEMBL4744310 0.86 SSTR4 (0.56) SSTR4HDAC3HDAC1HDAC2NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020260597-A1 COMPOSITIONS COMPRISING ENZYME CLEAVABLE LINKER PLATFORMS AND CONJUGATES THEREOF DANMARKS TEKNISKE UNIVERSITET (DK) 2020-12-30 WO disclosed
US-9266864-B2 VEGFR3 inhibitors CANCER THERAPEUTICS CRC PTY LIMITED (AU) 2016-02-23 US disclosed
US-9266864-B2 VEGFR3 inhibitors CANCER THERAPEUTICS CRC PTY LIMITED (AU) 2016-02-23 US disclosed
US-20150225377-A1 VEGFR3 INHIBITORS CANCER THERAPEUTICS CRC PTY LIMITED (AU) 2015-08-13 US disclosed
US-20150225377-A1 VEGFR3 INHIBITORS CANCER THERAPEUTICS CRC PTY LIMITED (AU) 2015-08-13 US disclosed
US-20140080798-A1 VEGFR3 INHIBITORS CANCER THERAPEUTICS CRC PTY LIMITED (AU) 2014-03-20 US disclosed
US-20140080798-A1 VEGFR3 INHIBITORS CANCER THERAPEUTICS CRC PTY LIMITED (AU) 2014-03-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150225377-A1 VEGFR3 INHIBITORS FLT4, FLT1, KDR SSTR4 610/4885HDAC3 4356/4885HDAC1 4357/4885
US-20140080798-A1 VEGFR3 INHIBITORS FLT4, FLT1, KDR SSTR4 508/4885HDAC3 3025/4885HDAC1 3331/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.