SCHEMBL15530516

SCHEMBL15530516

O=C(Nc1cccnn1)C1CNC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.41
GOT1 P17174 1/20 0.41
JAK2 O60674 2/20 0.40
FFAR2 O15552 1/20 0.40
GSK3B P49841 4/20 0.39
FAAH O00519 4/20 0.39
DYRK1A Q13627 3/20 0.39
FPR2 P25090 1/20 0.39
WNT1 P04628 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
ACVRL1 P37023 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HDAC2 Q92769 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
GSK3A P49840 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30751765 1.00 HPGD (0.47) HPGDSIRT2GOT1JAK2FFAR2
Hydrochloric Acid SCHEMBL21641085 0.98 HPGD (0.46) HPGDSIRT2GOT1JAK2FFAR2
SCHEMBL15530483 0.88 HPGD (0.46) HPGDSIRT2JAK2GSK3BFAAH
SCHEMBL8475732 0.79 NPC1 (0.56)
Hydrochloric Acid SCHEMBL30585989 0.78 NPC1 (0.54)
Hydrochloric Acid SCHEMBL21640960 0.78 NPC1 (0.54)
SCHEMBL29840665 0.75 CTSC (0.42) HPGDSIRT2GOT1JAK2FFAR2
SCHEMBL1734328 0.75 CTSC (0.42) HPGDSIRT2GOT1JAK2FFAR2
SCHEMBL5802284 0.75 TP53 (0.58) SMN1; SMN2
SCHEMBL1734935 0.74 SCN3A (0.46) HPGDGSK3BDYRK1AFPR2WNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2847181-A1 PYRIDAZINE AND PYRIDINE DERIVATIVES AS NAMPT INHIBITORS AbbVie Inc. (US) 2015-03-18 EP claimed
WO-2013170115-A1 PYRIDAZINE AND PYRIDINE DERIVATIVES AS NAMPT INHIBITORS ABBVIE INC. (US) 2013-11-14 WO claimed
EP-2847181-A1 PYRIDAZINE AND PYRIDINE DERIVATIVES AS NAMPT INHIBITORS AbbVie Inc. (US) 2015-03-18 EP disclosed
WO-2013170115-A1 PYRIDAZINE AND PYRIDINE DERIVATIVES AS NAMPT INHIBITORS ABBVIE INC. (US) 2013-11-14 WO disclosed