SCHEMBL1553394

SCHEMBL1553394

CCNC(=O)Nc1ncc(-c2cncc(C(=O)OCC)c2)cc1C(=O)OCC

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NAMPT P43490 4/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CHEK2 O96017 1/20 0.39
CDK8 P49336 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1553392 0.82 PIK3CD (0.48)
SCHEMBL1553271 0.81 CDK8 (0.42) KMT2AKDM4EMAPTCDK8
SCHEMBL1505706 0.80 KDM4E (0.43) CYP2C9CYP2C19POLBTSHRNPSR1
SCHEMBL1505581 0.80 KDM4E (0.43) CYP2C9CYP2C19NAMPTKMT2AGAA
SCHEMBL1505602 0.79 KDM4E (0.42) CYP2C9CYP2C19NAMPTKMT2AGAA
SCHEMBL13299066 0.77 PIK3CA (0.49)
SCHEMBL1552585 0.76 ABL1 (0.45) CYP2C9CYP2C19
SCHEMBL1553500 0.76
SCHEMBL1553061 0.76 ABL1 (0.47)
SCHEMBL1505580 0.75 CYP2C9 (0.43) CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2102199-B1 ANTIBACTERIAL POLYCYCLIC UREA COMPOUNDS ASTRAZENECA AB (SE) 2011-04-27 EP disclosed